Antiviral Mechanisms and Preclinical Evaluation of Amantadine Analogs that Continue to Inhibit Influenza A Viruses with M2 S31N-Based Drug Resistance
Ian Tietjen, Daniel Kwan, Annett Petrich, Roland Zell, Ivi Theodosia Antoniadou, Agni F. M. Gavriilidou, Christina Tzitzoglaki, Michail Christou Rallis, David Fedida, Francesc Xavier Sureda, Cato Mestdagh, Lieve M. J. Naesens, Salvatore Chiantia, F. Brent Johnson, Antonios Kolocouris
This study evaluates amantadine analogs against influenza A viruses with M2S31N resistance, finding some inhibit viral entry and assembly while being tolerated in mice.
Antiviral Research · Feb 11, 2025Peer-reviewedMicrobiology