Methionyl-tRNA synthetase inhibitor has potent in vivo activity in a novel Giardia lamblia luciferase murine infection model
S. A. Michaels, H.-W. Shih, B. Zhang, E. D. Navaluna, Z. Zhang, R. M. Ranade, J. R. Gillespie, E. A. Merritt, E. Fan, F. S. Buckner, A. R. Paredez, K. K. Ojo
The paper develops a luciferase-based murine model and cell assay to evaluate the efficacy of MetRS inhibitor 1717 against Giardia lamblia, showing its potent in vivo activity.
bioRxiv · Oct 29, 2019Microbiology