Pharmacology & ToxicologybioRxivPreprint
Targeting MYC Overexpressing Leukemia with Cardiac Glycoside Proscillaridin Through Downregulation of Histone Acetyltransferases
Elodie M. Da Costa, Gregory Armaos, Gabrielle McInnes…·Noël J-M Raynal
This study shows proscillaridin, a cardiac glycoside, selectively targets MYC overexpressing leukemia by downregulating histone acetyltransferases and inducing hematopoietic differentiation.
DOI 10.1101/444133