PP-2, a src-kinase inhibitor, is a potential corrector for F508del-CFTR in cystic fibrosis
Yunguan Wang, Kavisha Arora, Fanmuyi Yang, Woong‐Hee Shin, Jing Chen, Daisuke Kihara, Anjaparavanda P. Naren, Anil Goud Jegga
The paper identifies PP-2, a src-kinase inhibitor, as a novel corrector for ΔF508-CFTR in cystic fibrosis through in silico screening and experimental validation.
bioRxiv · Mar 24, 2018 · PreprintSystems Biology