BiochemistrybioRxiv
Using a fragment-based approach to identify novel chemical scaffolds targeting the dihydrofolate reductase (DHFR) from Mycobacterium tuberculosis
J. A. Ribeiro, A. Hammer, G. A. L. Zuniga…·M. V. B. Dias
This study uses fragment-based drug discovery to identify novel chemical scaffolds targeting Mycobacterium tuberculosis DHFR, revealing a new binding mode and low micromolar affinity compounds.
DOI 10.1021/acsinfecdis.0c00263