Non-blocking modulation contributes to sodium channel inhibition by a covalently attached photoreactive riluzole analog
P. Lukacs, M. C. Foldi, L. Valanszki, E. Casanova, B. Biri-Kovacs, L. Nyitray, A. Malnasi-Csizmadia, A. Mike
This study shows that non-blocking modulation of sodium channels is possible using a covalently attached photoreactive riluzole analog, suggesting new avenues for drug development.
bioRxiv · Dec 4, 2017Pharmacology & Toxicology