Pharmacology & ToxicologybioRxivPreprint
Preclinical Evaluation of a Novel BOC-Modified Triazoloacridinone (TRA-01AR) in Combination with 5-Fluorouracil in Colorectal Cancer
Marta Switalska, Paulina Czechowicz, Magdalena Milczarek…·Joanna Wietrzyk
This study evaluates the combination of 5-FU with two triazoloacridinones, C-1305 and TRA-01AR, in CRC, finding that C-1305 shows greater antitumor activity while TRA-01AR has improved tolerability and vascular effects.
DOI 10.64898/2026.11.08.765151