Harnessing Ionic Selectivity In Acetyltransferase Chemoproteomic Probes
Y. Jing, J. L. Montano, M. J. Levy, J. Lopez, P.-P. Kung, P. Richardson, K. Krajewski, L. Florens, M. Washburn, J. L. Meier
The paper develops a CoA-based chemoproteomic strategy to optimize probe selectivity and evaluates its application in assessing small molecule acetyltransferase inhibitors.
bioRxiv · Sep 24, 2020Biochemistry