Structural basis for stereospecific inhibition of ASCT2 from rational design
R.-A. A. Garibsingh, E. Ndaru, A. A. Garaeva, M. Bonomi, D. J. Slotboom, C. Paulino, C. Grewer, A. Schlessinger
The paper rationally designs inhibitors for ASCT2 using computational modeling and cryo-EM, showing how stereospecific pockets can be exploited for drug discovery.
bioRxiv · May 29, 2020Biochemistry