NeuroscienceJournal of Structural BiologyPeer-reviewed
Crystal structure of the GluK1 ligand-binding domain with kainate and the full-spanning positive allosteric modulator BPAM538
Yasmin Bay, Federico Míguez‐Cabello, Chloe C Koens…·J.S. Kastrup
The paper reports the crystal structure of the GluK1 ligand-binding domain complexed with kainate and the full-spanning positive allosteric modulator BPAM538, showing its unique binding mode and selectivity for GluK1.