A new chemotype of chemically tractable nonsteroidal estrogens based on a thienopyrimidine core.
V. R. Sammeta, J. D. Norris, S. Artham, C. D. Torrice, J. Byemerwa, C. Joiner, S. W. Fanning, D. P. McDonnell, T. M. Willson
The paper identifies a new chemotype of nonsteroidal estrogens based on a thienopyrimidine core through targeted screening and structure-guided optimization.
bioRxiv · Apr 15, 2022Cell Biology