NeuroscienceNeuropharmacologyPeer-reviewed
CHIR99021 causes inactivation of Tyrosine Hydroxylase and depletion of dopamine in rat brain striatum
Sally Hamdon, Pol Fernandez-Gonzalez, Muhammad Yusof Omar…·Carles Gil
This study shows CHIR99021 inhibits tyrosine hydroxylase and reduces dopamine in rat striatum, suggesting potential therapeutic use and caution in clinical trials.
3 citations