MicrobiologyAntimicrobial Agents and ChemotherapyPeer-reviewed
Characterization of antimalarial activity of artemisinin-based hybrid drugs
Helenita Costa Quadros, Lars Herrmann, Jeanne Manaranche…·Diogo Rodrigo Magalhães Moreira
This study characterizes the antimalarial activity of two artemisinin-based hybrid drugs against drug-sensitive and resistant Plasmodium falciparum parasites, finding that slow peroxide bond homolysis correlates with increased efficacy against resistant strains.
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