BiochemistrybioRxivPreprint
RAF isoform selectivity of MEK inhibitors and rational design of a covalent ARAF-MEK inhibitor
Sayan Chakraborty, Jie Jiang, Javier Viñals…·Michael J. Eck
The paper investigates MEK inhibitor selectivity across RAF isoforms and develops a covalent ARAF-MEK inhibitor with improved potency.