Pharmacology & ToxicologyNature CommunicationsPeer-reviewed
Steric control of signaling bias in the immunometabolic receptor GPR84
Pinqi Wang, Xuan Zhang, Akim Abdul Guseinov…·Angela J. Russell
The paper identifies ligands with varying steric profiles that exhibit different β-arrestin recruitment capacities at GPR84, revealing a mechanism for controlling signaling bias.
3 citations