Cell BiologybioRxivPreprint
A First-In-Class Broad Spectrum Inhibitor of Copper Exporting P1B-type ATPases
Vinit Shanbhag, Samuel Anakpeba-Dinguyella, Nikita Gudekar…·Michael J. Petris
This paper identifies MKV3 as the first small-molecule inhibitor of Cu+-transporting P1B-type ATPases, showing broad activity across species and defining a conserved Cu+ entry pocket for drug development.