Development of a dual chemical probe for the USP16 and HDAC6 zinc-finger ubiquitin-binding domain
Madhushika Silva, Mandeep Kaur Mann, Bijan Mirabi, Magdalena M. Szewczyk, Joachim Loup, Aurélien Dupeux, Renu Chandrasekaran, Jonathan Bajohr, C.H. Arrowsmith, Matthieu Schapira, Mark Lautens, Dalia Barsyte-Lovejoy, Rachel Harding, Vijayaratnam Santhakumar
The paper develops a chemical probe targeting the USP16 zinc-finger ubiquitin-binding domain and evaluates its selectivity and activity in cellular assays.
Journal of Medicinal Chemistry · Feb 20, 2026Peer-reviewedMolecular Biology