Molecular BiologyJournal of Medicinal ChemistryPeer-reviewed
Structure-guided design and optimization of covalent VHL-targeted sulfonyl fluoride PROTACs
Rishi R. Shah, Elena De Vita, Preethi Soundarya Sathyamurthi…·Edward W. Tate
This study designs and optimizes covalent VHL-targeted sulfonyl fluoride PROTACs that degrade BRD4 and androgen receptor without linker optimization.
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