Structure-Activity Relationship Studies Towards Analogues of Pleconaril as Novel Enterovirus-D68 Capsid-Targeting Antivirals
David L. Cousins, Ed Griffen, Jessica Stacey, Alpha A. Lee, Yuliia Filimonova, Anton Hlavin, Yuliia Holota, Roman Khmil, Mykyta V. Kordubailo, Oleksii Kostinov, Dmytro S. Lesyk, Ivan G. Logvinenko, Mariia Lototska, Viacheslav Lysenko, A. Pashchenko, , Kris M. White
The paper investigates structure-activity relationships of pleconaril analogues against EV-D68, identifying compounds with antiviral activity and favorable ADME properties.
bioRxiv · Aug 8, 2025 · PreprintPharmacology & Toxicology