MicrobiologybioRxivPreprint
Discovery of ARQ-501 as a potent PafA inhibitor that elevates KatG levels to potentiate isoniazid in mycobacteria
Cong Li, Bingzhou Huang, Hang Xiong…·Qingxiang Sun
The paper identifies ARQ-501 as a PafA inhibitor that increases KatG levels, enhancing isoniazid efficacy against tuberculosis.
DOI 10.64898/2026.06.03.729796