Pharmacology & ToxicologyACS Medicinal Chemistry LettersPeer-reviewed
Lysineless HiBiT and NanoLuc Tagging Systems as Alternative Tools Monitoring Targeted Protein Degradation
Hanfeng Lin, Kristin M. Riching, May Poh Lai…·Jin Wang
This study introduces lysineless HiBiT-RR and nLucK0 tagging systems to reduce degradation artifacts in monitoring protein degradation, showing HiBiT-RR retains sensitivity and nLucK0 shows different degradation patterns than nLucWT.
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