Cancer BiologybioRxivPreprint
CDK12/13 inhibitor, CTX-439, suppresses tumor growth and potentiates BCL-2 family blockade
Hiroko Yamakawa, Raghda Khatab, Akio Mizutani…·Kosuke Yusa
This study develops CTX-439, a CDK12/13 inhibitor, showing anti-tumor effects and resistance mechanisms, and proposes combining it with BCL-2 family inhibitors for cancer treatment.
2 citations