Pharmacology & ToxicologyAngewandte Chemie International EditionPeer-reviewed
A Kinetic Scout Approach Accelerates Targeted Protein Degrader Development
Angela T. Fan, Gillian E. Gadbois, Hai‐Tsang Huang…·Fleur M. Ferguson
This study develops a kinetic scout approach to accelerate targeted protein degrader development by tuning ligand residence time through chemical proteomics and mechanistic assays.
10 citations