BiochemistryJournal of the American Chemical SocietyPeer-reviewed
A Functional Assay For Mining Non-Inhibitory Enzyme Ligands From One Bead One Compound Libraries: Application to E3 Ubiquitin Ligases
Weijun Gui, Allison Goss, Thomas J. Kodadek
The paper introduces a functional assay to identify non-inhibitory enzyme ligands from bead-displayed compound libraries, applied to E3 ubiquitin ligases, and discovers a novel ligand for VHL.