Vector-Mediated Transport Producing Drug-like Peptides
K. A. Gruber, J. A. Cowan, A. Cowan, W. Qi, S. Pearson, M. J. Ross, C. Wachnowsky, F. Gallazzi, S. Jiang, S. R. Van Doren, M. F. Callahan
This paper develops a vector-mediated transport approach to create drug-like peptides with oral activity, blood-brain-barrier transport, and extended in vivo half-life.
bioRxiv · Dec 28, 2018 · PreprintPharmacology & Toxicology