Structural insights into the agonist selectivity and structure-based engineering of the adenosine A3 receptor
Hidetaka S. Oshima, Akiko Ogawa, Fumiya K. Sano, Hiroaki Akasaka, Tomoyoshi Kawakami, Aika Iwama, Hiroyuki H. Okamoto, Chisae Nagiri, Fan‐Yan Wei, Wataru Shihoya, Osamu Nureki
The paper identifies a novel A3R-selective ligand and reveals structural insights into A3R activation, enabling structure-guided engineering of m6A-insensitive A3R for drug discovery.
Nature Communications · Nov 7, 2024Peer-reviewedBiophysics