BiochemistrybioRxiv
Molecular insights into intrinsic transducer-coupling bias in the CXCR4-CXCR7 system
P. Sarma, H.-J. Yoon, C. M. Carino…·A. K. Shukla
This study characterizes the biased agonism of CXCR4 and CXCR7, revealing differences in G-protein coupling, β-arrestin recruitment, and ERK1/2 activation.
DOI 10.1038/s41467-023-40482-9