FCD-11: A First-in-Class COMPASS Inhibitor in Cancer Therapeutics
Zibo Zhao, Meenal Karunanidhi, Sarah R. Gold, Luke St John, Rukkia Liaqat, Marta Iwanaszko, Claudia Bigas, Eita Uchida, Kentaro Mineji, Jun Watanabe, Salvador Aznar-Benitah, Rintaro Hashizume, Rama K. Mishra, Ali Shilatifard
The paper identifies and characterizes FCD-11, a first-in-class COMPASS inhibitor that reduces tumor size and extends survival in breast cancer models.
bioRxiv · Jul 31, 2026 · PreprintBiochemistry