Design and Synthesis of Potent First-in-Class Histones Acetyltransferase Modulators.
Elisa Zuccarello, Mattia Mori, Elisa Calcagno, Rosa Purgatorio, Yan Feng, Erica Acquarone, Yitshak I. Francis, Mauro Fà, Agnieszka Staniszewski, Elentina K. Argyrousi, Coleman D. Barry, Hong Zhang, Shi-Xian Deng, Donald W. Landry, Ottavio Arancio, Jole Fiorito
The paper designs and synthesizes new activators of the p300 histone acetyltransferase enzyme to treat neurodegenerative and cancer disorders.
bioRxiv · Mar 3, 2025 · PreprintBiochemistry