Structure Activity Relationship of USP5 Allosteric Inhibitors
M. K. Mann, C. A. Zepeda-Velazquez, H. G. Alvarez, A. Dong, T. Kiyota, A. Aman, C. Arrowsmith, R. Al-Awar, R. J. Harding, M. Schapira
This paper develops a chemical series of USP5 allosteric inhibitors, identifies a selective compound with structural and functional characterization.
bioRxiv · May 17, 2021 · PreprintBiochemistry