Chromomycin A2 potently inhibits glucose-stimulated insulin secretion from pancreatic β cells.
M. A. Kalwat, I. H. Hwang, J. Macho, M. G. Grzemska, J. Z. Yang, K. McGlynn, J. B. MacMillan, M. H. Cobb
This study identifies chromomycin A2 as a potent inhibitor of glucose-stimulated insulin secretion from pancreatic β cells through multiple mechanisms including Wnt signaling disruption and calcium influx suppression.
bioRxiv · Jul 10, 2018Cell Biology