Pharmacology & ToxicologybioRxiv
Receptor levels determine binding affinity of WNT-3A to Frizzled 7 in a colorectal cancer model
L. Graetz, J. J. Sajkowska-Kozielewicz, J. Wesslowski…·P. Kozielewicz
The paper assesses WNT-3A binding affinity to endogenous versus overexpressed FZD7 in colorectal cancer cells and finds lower affinity with higher receptor concentrations.
DOI 10.1111/bph.16090