Cancer BiologyMoleculesPeer-reviewed
Biguanide-PROTACs: Modulating Mitochondrial Proteins in Pancreatic Cancer Cells
Julie Vatté, Véronique Bourdeau, Gerardo Ferbeyre, Andreea R. Schmitzer
This study synthesizes Biguanide-PROTACs and evaluates their activity on pancreatic cancer cells, finding structure-permeability-activity relationships and some AMPK activation.