Pharmacology & ToxicologybioRxiv
Orally Bioavailable Endochin-like Quinolone Carbonate Ester Prodrug Reduces Toxoplasma gondii Brain Cysts
J. S. Doggett, T. L. Schultz, A. Miller…·V. B. Carruthers
This study develops an orally bioavailable prodrug of ELQ-316 that enhances its plasma concentrations and efficacy against Toxoplasma gondii infection.
DOI 10.1128/aac.00535-20