Pharmacology & ToxicologyActa Pharmaceutica Sinica BPeer-reviewed
A neurotensin receptor type 1-derived pepducin acts as a biased allosteric modulator to regulate target receptor function
Rebecca L. Brouillette, Frédérique Lussier, Émile Breault…·Philippe Sarret
This paper describes a pepducin derived from NTS1 that acts as a biased allosteric modulator, preferentially activating G proteins over β-arrestin and inhibiting receptor internalization.
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