Covalent Inhibition of New Delhi Metallo-β-Lactamases NDM-1 and NDM-5 by 3-Bromopyruvate
Jack K. Bradley, Karina Calvopiña, Sabrina J. Moyo, Ellinor Shore, Peter Nambala, W. David Hong, Christopher Joseph Schofield, Adam Paul Roberts
This study shows 3-BP covalently inhibits NDM-1 and NDM-5 MBLs, restoring carbapenem activity against resistant bacterial strains.
JAC-Antimicrobial Resistance · Jul 2, 2026Peer-reviewedMicrobiology