TRPV4 Inhibition by a Natural Product Mediates Analgesia
Zhen Yuan, Jie Qiu, Shiliang Li, Hanqing Zhao, Na Chen, Shanshan Ruan, Yu Gan, Jiawen Wang, Tianyu Ye, Wenjie Liao, Ziyuan Li, Yanyan Diao, Lili Zhu, Zhenjiang Zhao, Rui Wang, , Bowen Ke
This study identifies AH001 as a potent TRPV4 inhibitor, revealing its mechanism and demonstrating its analgesic effects in pain models.
bioRxiv · Jan 5, 2026 · PreprintBiochemistry