Pharmacology & ToxicologyCommunications BiologyPeer-reviewed
Structure-guided development of a potent human B0AT1 inhibitor effective in a mouse model of phenylketonuria
Takuya Imazu, Tomoya Akashi, Masahiro Hiraizumi…·Ikuko Miyaguchi
This study develops a potent B0AT1 inhibitor effective in a PKU mouse model by targeting an allosteric site.