Pharmacology & ToxicologyActa Pharmaceutica Sinica BPeer-reviewed
Primulagenin A is a potent inverse agonist of the nuclear receptor RAR-related orphan receptor gamma (RORγ)
Patrik F. Schwarz, Alexander F. Perhal, Teresa Preglej…·Verena Maria Dirsch
This study identifies primulagenin A as a potent inverse agonist of RORγ, showing efficacy in inhibiting Th17 cell differentiation and reducing IL-17A production.