CXCR1 and CXCR2 display receptor bias for shared chemokine agonists
Chanpreet Jassal, Joseph Strawn, Emily K. Walsh, Krishna Rajarathnam, Sudarshan Rajagopal
The paper shows that CXCL1 acts as a G protein-biased partial agonist at CXCR1 but a balanced full agonist at CXCR2, revealing receptor bias in chemokine signaling.
Molecular Pharmacology · Mar 5, 2026Peer-reviewedBiochemistry