BiochemistryMolecular PharmacologyPeer-reviewed
CXCR1 and CXCR2 display receptor bias for shared chemokine agonists
Chanpreet Jassal, Joseph Strawn, Emily K. Walsh…·Sudarshan Rajagopal
The paper shows that CXCL1 acts as a G protein-biased partial agonist at CXCR1 but a balanced full agonist at CXCR2, revealing receptor bias in chemokine signaling.
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