Pharmacology & ToxicologybioRxivPreprint
Structure-Guided Design of C5aR1-Selective Peptide Agonists
Joshua C Dent, Xiaosa Wu, Liam Rogl, Richard J. Clark
This study designs C5aR1-selective peptide agonists using structure-guided computational methods and experimental validation, showing improved selectivity and stability through specific amino acid substitutions.
DOI 10.64898/2026.09.02.746116