Pharmacology & ToxicologybioRxivPreprint
Antimuscarinic drugs exert β-arrestin-biased agonism at the muscarinic acetylcholine type 1 receptor
Shayan Amiri, Mohamad‐Reza Aghanoori, Darrell R. Smith…·Paul Fernyhough
Antimuscarinic drugs act as β-arrestin-biased agonists via casein kinase 2 activation to promote ERK1/2 phosphorylation and neurite outgrowth.
DOI 10.1101/2025.04.16.649213