Development of radiofluorinated MLN-4760 derivatives for PET imaging of the SARS-CoV-2 entry receptor ACE2
Jinling Wang, Darja Beyer, Christian Vaccarin, Yingfang He, Matthias Tanriver, Roger Benoit, Xavier Deupí, Linjing Mu, Jeffrey W. Bode, Roger Schibli, Cristina Müller
This paper develops and evaluates radiofluorinated derivatives of MLN-4760 for PET imaging of ACE2, finding that [18F]F-MLN-4760 shows superior binding affinity and yield.
European Journal of Nuclear Medicine and Molecular Imaging · Jul 27, 2024Peer-reviewedPharmacology & Toxicology