Effective Tubulin Degradation by Rationally Designed Proteolysis Targeting Chimeras
Alice Maiocchi, Anne‐Catherine Abel, Milo Jarno Basellini, Helena Pérez‐Peña, Zlata Boiarska, Erica Elisa Ferrandi, Zuzanna Kozicka, Valerio Fasano, Stefano Pieraccini, Graziella Cappelletti, Michel Olivier Steinmetz, Daniele Passarella, Andrea Enrico Prota
This study designs and tests PROTACs targeting β-tubulin, showing two compounds effectively degrade tubulin in cells.
bioRxiv · May 22, 2025 · PreprintBiochemistry