Cancer BiologybioRxivPreprint
A bivalent lysine-acetylated small-molecule binding site in MYC
Dikshat Gopal Gupta, Mihai Ioan Truica, Jin‐gon Shim…·Sarki Abba Abdulkadir
This study identifies a bivalent binding site in MYC for small-molecule inhibitors and shows acetylation enhances inhibitor binding and oncogenic activity.
DOI 10.64898/2026.03.02.707789