BiochemistryBioorganic & Medicinal Chemistry LettersPeer-reviewed
Synthesis of K+ channel radioligand 5-methyl-3-fluoro-4-aminopyridine and PET imaging in mice
Yang Sun, Karla M. Ramos‐Torres, Kazue Takahashi…·Pedro Brugarolas
This paper synthesizes [18F]5Me3F4AP, a K+ channel PET radioligand, and demonstrates its brain uptake and kinetics in mice, suggesting it as a potential improved tracer for demyelination imaging.