NeurosciencebioRxivPreprint
Dizocilpine-derived K2060 exhibits enhanced blockage at NMDA receptors with impaired Mg2+ block and provides strong protection against audiogenic seizures
Marharyta Kolcheva, Jakub Netolický, Anna Misiachna…·Martin Hořák
This study evaluates how impaired Mg2+ block at NMDA receptors affects the efficacy of K2060, memantine, and ketamine in protecting against audiogenic seizures.
DOI 10.64898/2026.10.06.756690