NeurosciencebioRxivPreprint
A Small-molecule Antagonist Radiotracer for Positron Emission Tomography Imaging of the Mu Opioid Receptor.
Konstantinos Plakas, Chia‐Ju Hsieh, Dinahlee Saturnino Guarino…·Robert H. Mach
This paper designs and characterizes non-agonist ligands for the mu opioid receptor, identifies a radiotracer [11C]1A for PET imaging, and demonstrates its brain uptake and receptor specificity in rhesus macaques.
1 citation