BiochemistryRSC Medicinal ChemistryPeer-reviewed
Electrostatic interactions define nacubactam potency against OXA-48-like β-lactamases
Joseph F. Hoff, Kirsty E. Goudar, Karina Calvopiña…·JAMES M. SPENCER
This paper compares the potency of nacubactam and avibactam against OXA-48-like β-lactamases, finding that nacubactam is less potent due to electrostatic repulsion with Arg214.